Drugs used in the treatment of asthma Classification in Grash Course: Respiratory system(2nd Edition) a Relievers Bronchodilators P2 agonists short-acting: salbutamol, terbutaline long-acting: salmeterol, formoterol Anticholinergics(muscarinic antagonists): ipratropine Xantines(theophyllines): aminophylline a Preventers- Anti-inflammatory drugs Glucocorticosteroids: Inhaled steroids: beclomethasone, budesonide, fluticasone oral steroids: hydrocortisone, prednisone, dexamethasone Leukotriene(LT) receptor antagonists (leukotriene modifiers) LT antagonists: montelukast(孟鲁司特), zafirlukast(扎鲁司特 5- lipoxygenase inhibitors: zileuton(齐留通 Inhibitors of mediator release: cromolyn sodium, nedocromil
Drugs used in the treatment of asthma - Classification in Grash Course: Respiratory system (2nd Edition) -
Antiasthmatic drugs Glucocorticosteroids Systemic hydrocortisone氩化可的松 prednisone波尼松 dexamethasone地塞米松 Inhaled: beclomethasone dipropionate二丙酸倍氯米松 budesonide布地奈德 triamcinolone acetonide曲安奈德 fluticasone propionate丙酿酸氟普卡松 flunisolide尼缩松
Antiasthmatic drugs
Adrenocorticoid drugs Adrenocortical hormones MG neralocorticoids lucocorticoids "(Glucocorticosteroids) 冷 Sex hormones
Adrenocorticoid drugs vAdrenocortical hormones v Mineralocorticoids v Glucocorticoids v (Glucocorticosteroids) v Sex hormones
条经 Zona Glomerulosa P450 aldo AⅡ Aldosterone K ACTH P450 Zonae 11B Fasciculata/ P450 170 Reticularis Cortisol Androgens Medulla &2a careEN OSE
A. Glucocorticoid drugs 1. Pharmacological effects Mechanisms of glucocorticoid actions (1) Effects on metabolisms .(2 Permissive action (3)Anti-inflammatory effects (4)Effects on immune and allergy ( 5)Anti-shock (6Other effects antipyretic effects effects on blood and blood-forming organs skeletal system CNS effects
A. Glucocorticoid drugs