Medicinal Chemistry Chapter 3 Peripheral Nervous System Drugs
Medicinal Chemistry Chapter 3 Peripheral Nervous System Drugs
Outline Drug Affecting Cholinergic Cholinergic Drugs Neurotransmission Anticholinergic drugs Drug Affecting Adrenergic+ Adrenergic Drugs(agonist Neurotransmission Adrenergic Antagonist (Chapter 4) Antihistamines Histamine H, Receptor Antagonists Local Anesthetics
Outline Drug Affecting Cholinergic Neurotransmission Cholinergic Drugs Anticholinergic Drugs Drug Affecting Adrenergic Neurotransmission Adrenergic Drugs (agonist) Adrenergic Antagonist (Chapter 4) Antihistamines Histamine H1 Receptor Antagonists Local Anesthetics
3.1 Cholinergic Drugs(拟胆碱药) ° Cholinergic effect Mediated by acetylcholine (ACh) N Acetylcholine
3.1 Cholinergic Drugs (拟胆碱药) • Cholinergic effect Mediated by acetylcholine (ACh)
Biosynthesis of acetylcholine Serine Choline COoH decarboxylase N-methyltransferase NH. HO )NH2 Choline acetyltransferase AcylCholine
Biosynthesis of Acetylcholine
The Classification of Cholinergic Drugs Cholinoceptor agonists Cholinergic Drugs Acetylcholinesterase inhibitors (AChEIs
The Classification of Cholinergic Drugs Acetylcholinesterase inhibitors (AChEIs) Cholinocepter agonists Cholinergic Drugs